Overview

MOTS-c is a 16-amino acid mitochondrial-derived peptide (MDP) encoded by a short open reading frame within the 12S rRNA gene of mitochondrial DNA. It is one of the most recently discovered endogenous peptide hormones, identified in 2015, and functions as a regulator of metabolic homeostasis and aging. Plasma MOTS-c levels decline ~21% by ages 70-81 compared to young adults, and exogenous MOTS-c treatment has demonstrated remarkable metabolic rescue effects in aging and obese models including prevention of diet-induced and age-related insulin resistance.

Mechanism of Action

MOTS-c translocates to the nucleus under metabolic stress, where it acts as a nuclear regulatory peptide influencing gene expression related to metabolism and stress response. Key mechanisms include: AMPK pathway activation driving metabolic flexibility; elevation of intracellular NAD+ levels through effects on the folate/methionine cycle; SIRT1 activation mediating glycolytic effects; restriction of methionine metabolism (methionine restriction extends mouse lifespan by 45%); reduction of IL-6-driven MMP1 in skin improving collagen retention; and enhancement of physical performance and insulin-sensitive tissue function.

Potential Benefits

  • Prevention and reversal of diet-induced obesity and insulin resistance
  • Prevention of postmenopausal obesity and metabolic syndrome
  • Improved physical performance across all age groups in animal models
  • Elevated NAD+ levels supporting cellular energy and longevity
  • AMPK activation mimicking exercise benefits metabolically
  • Cardiovascular disease risk reduction in aging models
  • Skin collagen preservation via IL-6/MMP1 reduction
  • Potential Alzheimer's disease and osteoporosis protection

Dosage Protocols

The following reflects doses used in published research studies. This is not medical advice. Consult a qualified healthcare professional.

Typical Range5-10 mg/week
Beginner5 mg once weekly
Intermediate5-10 mg twice weekly
Advanced10 mg 2-3x/week
Cycle Duration4-8 weeks
Cycle Off4 weeks

MOTS-c is mitochondria-derived and endogenously increases with exercise. Exogenous administration mimics exercise-induced metabolic adaptation. Best combined with physical exercise for synergistic metabolic benefits.

Routes of Administration

Subcutaneous Injection High

Primary research route; systemic delivery for metabolic and exercise-mimetic effects

Intramuscular Injection High

Alternative; may be preferred for direct muscle metabolic targeting

Stacking Protocols

Popular research stacks involving MOTS-c:

Mitochondrial Health Stack

Comprehensive mitochondrial optimization, energy production, and cellular survival

MOTS-c activates AMPK and biogenesis; SS-31 protects cardiolipin; Humanin reduces apoptosis; NAD+ provides substrate for sirtuins and PARP.

Metabolic + Longevity Stack

Exercise-mimetic metabolic benefits with anti-aging tissue repair

Suitable for older adults seeking metabolic improvement and longevity support without high-intensity exercise capacity.

Reconstitution

Typical Vial Size5mg, 10mg
BAC Water1-2ml per 5mg vial
StorageRefrigerate at 2-8°C after reconstitution
Shelf Life28 days refrigerated

Need exact syringe measurements?

Amino Acid Sequence

MRWQEMGYIFYPRKLR (16 amino acids)

Side Effects & Safety

  • Minimal known side effects in rodent studies
  • Limited human safety data
  • Injection site reactions with subcutaneous use

Synergistic Compounds

The following compounds have been studied alongside MOTS-c for potential complementary or synergistic effects:

SS-31HumaninNAD+ precursors (NMN, NR)5-Amino-1MQ

Learn More

References & Further Reading

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